Organocatalytic enantioselective direct vinylogous michael addition of α,β-unsaturated γ-butyrolactam to β-acyl acrylates and 1,2-diacylethylenes.

DOI Number:

10.1021/jo5027047

Reaction Category:

RXNO ID:

RXNO_0000009

Educt:

β-acyl acrylates, 1,2-diacylethylenes, α,β-unsaturated γ-butyrolactam

Product:

substituted (R)-2-((R)-5-oxo-2,5-dihydro-1H-pyrrol-2-yl)succinaldehyde

Catalyst:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(9R)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-25-8

Associated Product from Buchler GmbH:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(9R)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-25-8