Streocontrolled construction of six vicinal stereogenic centers on spiropyrazolones via organocascade Michael/Michael/1, 2-addition reactions.

DOI Number:

10.1021/ol501093v

Reaction Category:

Educt:

ethyl 3-oxobutanoate, (E)-(2-nitrovinyl)benzene, (Z)-4-benzylidene-5-methyl-2-phenyl-2,4-dihydro-3H-pyrazol-3-one

Product:

spiropyrazolones

Catalyst:

3-[[[3,5-Bis(trifluoromethyl)phenyl]methyl]amino]-4-[[(8α,9S)-6′-methoxycinchonan-9-yl]amino]-3-Cyclobutene-1,2-dione

Cas No:

1210360-60-3

Cas No:

130-95-0