A bifunctional squaramide-catalysed enantioselective vinylogous Michael addition/cyclization cascade reaction of 4-unsaturated isoxazol-5-ones and α,α-dicyanoalkenes.

DOI Number:

10.1039/D1OB01256H

Reaction Category:

Educt:

4-unsaturated isoxazol-5-ones, α,α-dicyanoalkenes

Product:

substituted (R)-6-imino-1-oxo-2-oxa-3-azaspiro[4.5]deca-3,7-diene-7-carbonitrile

Catalyst:

3-[[(8α,9S)-6′-methoxycinchonan-9-yl]amino]-4-[[4-(trifluoromethyl)phenyl]amino]-3-cyclobutene-1,2-dione

Cas No:

1256245-85-8

Cas No:

130-95-0