Stereoselective mechanochemical synthesis of thiomalonate Michael adducts via iminium catalysis by chiral primary amines.

DOI Number:

10.3762/bjoc.20.198

Reaction Category:

RXNO ID:

RXNO_0000009

Educt:

cyclohexenone, thiomalonates

Product:

S,S-dibenzyl (S)-2-(3-oxocyclohexyl)propanebis(thioate)

Catalyst:

2-fluorobenzoic acid, (8α,9S)-6′-Methoxycinchonan-9-amine

Cas No:

168960-95-0

Cas No:

130-95-0