Highly enantioselective conjugate addition of malononitrile to 2-enoylpyridines with bifunctional organocatalyst.

DOI Number:

10.1021/ol3015607

Reaction Category:

RXNO ID:

RXNO_0000009

Educt:

2-enoylpyridines, malononitrile

Product:

1-substituted 2-(3-oxo-3-(pyridin-2-yl)propyl)malononitrile

Catalyst:

N-[3,5-bis(trifluoromethyl)phenyl]-N′-(9R)-cinchonan-9-yl-urea

Cas No:

945985-98-8

Cas No:

118-10-5