Highly Enantioselective Monofluoromethylation of C2-Arylindoles Using FBSM under Chiral Phase-Transfer Catalysis.
DOI Number:
10.1021/ol4013102
Reaction Category:
MOP ID:
MOP_0000553
Educt:
2-aryl-3-(1-arylsulfonylmethyl)indoles, 1-fluoro-1,1-bis(phenylsulfonyl)methane
Product:
2-aryl-3-(2-fluoro-2,2-bis(phenylsulfonyl)ethyl)indoles
Catalyst:
1-[[3,5-bis(1,1-dimethylethyl)phenyl]methyl]-9-hydroxy-(9S)-Cinchonanium bromide (1:1)
Cas No:
1190864-60-8
Associated Product from Buchler GmbH:
Cinchonine Base
Cas No:
118-10-5