Highly Enantioselective Synthesis of γ-Carboxy-β-amino Acids via Desymmetric Alcoholysis of 3-Aminoglutaric Anhydrides.

DOI Number:

10.1021/acs.orglett.5c00955

Reaction Category:

Educt:

3-aminoglutaric anhydrides, methanol

Product:

γ-carboxy-β-amino acids

Catalyst:

3,4-Bis[[(8α,9S)-6′-methoxycinchonan-9-yl]amino]-3-cyclobutene-1,2-dione

Cas No:

1204591-48-9

Cas No:

130-95-0