Organocatalytic Asymmetric One-Step Desymmetrizing Dearomatization Reaction of Indoles: Development and Bioactivity Evaluation.

DOI Number:

10.1002/anie.201811437

Reaction Category:

MOP ID:

MOP_0000561

Educt:

substituted 1-((2-((1H-indol-3-yl)methyl)phenyl)ethynyl)naphthalen-2-ol

Product:

substituted (5aR,10aR)-10,10a-dihydro-5H-benzo[5,6]naphtho[2',3':3,4]chromeno[2,3-b]indole

Catalyst:

N-[3,5-bis(trifluoromethyl)phenyl]-N′-(9R)-cinchonan-9-yl-thiourea

Cas No:

851477-19-5

Cas No:

118-10-5