Diastereo-and Enantioselective Synthesis of Functionalized Cyclopentenes Containing a Quaternary Chiral Center via a Thiosquaramide-Catalyzed Cascade Michael–Henry Reaction.

DOI Number:

10.1021/acs.joc.9b02176

Reaction Category:

RXNO ID:

RXNO_0000086

Educt:

substituted 2-(2-oxoethyl)malononitrile, (E)-1-nitroalk-1-enes

Product:

2,4-disubstituted (1S,2R)-1-cyano-3-nitrocyclopent-3-ene-1-carboxamide

Catalyst:

3-[[(9R)-6′-methoxycinchonan-9-yl]amino]-4-[(phenylmethyl)amino]-3-cyclobutene-1,2-dithione

Cas No:

2390162-31-7

Cas No:

56-54-2