Highly enantioselective amination reactions of fluorinated keto esters catalyzed by novel chiral guanidines derived from cinchona alkaloids.

DOI Number:

10.1002/adsc.201000562

Reaction Category:

Educt:

fluorinated keto esters, di‐tert‐butyl azodicarboxylate

Product:

diethyl (R)-1-(2-fluoro-1-methoxy-1,3-dioxo-3-phenylpropan-2-yl)hydrazine-1,2-dicarboxylate

Catalyst:

N-[3,5-bis(trifluoromethyl)phenyl]-N′-[(9R)-6′-methoxycinchonan-9-yl]-guanidine

Cas No:

1260109-05-4

Cas No:

56-54-2