C60 steric bulk of cinchona alkaloid enables an enantioselective Michael addition/annulation sequence toward pyranopyrazoles.

DOI Number:

10.1039/c8cc00154e

Reaction Category:

MOP ID:

MOP_0000561

Educt:

2-(phenylethynyl)cyclohex-2-en-1-one, 2,5-diphenyl-2,4-dihydro-3H-pyrazol-3-one

Product:

(S)-5-benzyl-1,3-diphenyl-7,8,9,9a-tetrahydroisochromeno[3,4-c]pyrazol-6(3H)-one

Catalyst:

(8α,9R)-6′-[[Tris(1-methylethyl)silyl]oxy]cinchonan-9-ol

Cas No:

876269-53-3

Cas No:

524-63-0