Bifunctional Thiourea-Catalyzed Enantioselective Aza-Friedel–Crafts Reaction of 3-Aminobenzofurans with Isatin-Derived Ketimines.

DOI Number:

10.1021/acs.joc.3c01741

Reaction Category:

RXNO ID:

RXNO_0000369

Educt:

3-aminobenzofurans, isatin-derived ketimines

Product:

substituted tert-butyl (R)-(3-(3-aminobenzofuran-2-yl)-2-oxoindolin-3-yl)carbamate

Catalyst:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(8α,9S)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-16-7

Cas No:

130-95-0