Catalytic enantioselective hydrophosphinylation of in situ-generated indole-derived vinylogous imines to access 3-(1-diphenylphosphoryl-arylmethyl) indoles.

DOI Number:

10.1039/d2cc04763b

Reaction Category:

Educt:

2-methyl-3-(phenyl(tosyl)methyl)-1H-indole, bis(4-(trifluoromethyl)phenyl)phosphine oxide

Product:

(S)-((2-methyl-1H-indol-3-yl)(phenyl)methyl)bis(4-(trifluoromethyl)phenyl)phosphine oxide

Catalyst:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(8α,9S)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-16-7

Associated Product from Buchler GmbH:

N-[3,5-Bis(trifluoromethyl)phenyl]-N′-[(8α,9S)-6′-methoxycinchonan-9-yl]thiourea

Cas No:

852913-16-7